-
María Fuertes, Asier Selas, Angela Trejo, Birgitta R. Knudsen, Francisco Palacios, Concepción Alonso
Synthesis of hybrid phosphorated indenoquinolines and biological evaluation as topoisomerase I inhibitors and antiproliferative agents
Bioorganic & Medicinal Chemistry Letters,
2022;
57,
128517 - 128524 -
0960-894X
-
Ann-Katrine Jakobsen, Josephine Geertsen Keller, M. Gonzalez, E. Martin-Encinas, F. Palacios, C. Alonso, Birgitta R. Knudsen, Magnus Stougaard
A Dual-Sensor-Based Screening System for In Vitro Selection of TDP1 Inhibitors
Sensors,
2021;
21,
4832 - 4848
-
A. Selas, E. Martin-Encinas, M. Fuertes, C. Masdeu, C. Rubiales, F. Palacios, C. Alonso
A Patent review of topoisomerase I inhibitors (2016 – present)
Expert Opinion on Therapeutic Patents,
2021;
31,
473 - 508
-
A. Selas, G. Ramirez, , F. Palacios, C. Alonso
Design, synthesis and cytotoxic evaluation of diphenyl(quinolin-8-yl)phosphine oxides
Tetrahedron Letters,
2021;
70,
153019 - 153023
-
A. Selas M. Fuertes, E. Melcón-Fernández, Y. Pérez-Pertejo, R. M. Reguera, R. Balaña-Fouce,, B. R. Knudsen, F. Palacios, and C. Alonso
Hybrid Quinolinyl Phosphonates as Heterocyclic Carboxylate Isosteres: Synthesis and Biological Evaluation against Topoisomerase 1B (TOP1B)
Pharmaceuticals,
2021;
14,
784 - 908
-
E. Martin-Encinas, G. Rubiales, B. R. Knudssen, F. Palacios, C. Alonso
Fused chromeno and quinolino[1,8]naphthyridines: Synthesis and biological evaluation as topoisomerase I inhibitors and antiproliferative agents
Bioorganic Medicinal Chemistry,
2021;
40,
116177 - 116192
-
F. Palacios, A. M. Ochoa de Retana, J. M. de los Santos
Copper in N-Heterocyclic Chemistry
Copper in N-Heterocyclic Chemistry,
2021;
1 - 44 -
978-0-12-821263-9
-
Kamilla Vandsø Petersen, Asier Selas, Kirstine Mejlstrup Hymøller, Karol Mizielinski, Maria Thorsager, Magnus Stougaard, Conception Alonso, Francisco Palacios, Yolanda Perez Pertejo, Rosa Maria Reguera, Rafael Balana Fouce, Birgitta R. Knudsen, Cinzia Tesauro
Simple and Fast DNA Based Sensor System for Screening of Small-molecule compounds Targeting Eukaryotic Topoisomerase1
Pharmaceutics,
2021;
13 - 1255 -
1270
-
M. Jewginski, K. Haremza , J. M. de los Santos , Z. Es Sbai, B. Oszywa, M. Pawelczak, F. Palacios, R. Latajka
Phosphinotripeptidic inhibitors of leucylaminopeptidases
International Journal of Molecular Sciences,
2021;
22,
5090 - 5117
-
V. Carramiñana, Ana M. Ochoa de Retana, F. Palacios, J M de los Santos
Synthesis and antiproliferative activity of phosphorus substituted 4-cyanooxazolines, 2-aminocyano oxazoliines, 2-iminocyanooxazolidines and 2-aminocyanothiazolines by rearrangement of cyanoaziridines
Molecules,
2021;
26,
4265 - 4292