-
María Fuertes, Asier Selas, Angela Trejo, Birgitta R. Knudsen, Francisco Palacios, Concepción Alonso
Synthesis of hybrid phosphorated indenoquinolines and biological evaluation as topoisomerase I inhibitors and antiproliferative agents
Bioorganic & Medicinal Chemistry Letters,
2022;
57,
128517 - 128524 -
0960-894X
-
X. del Corte; A. López-Francés, E. Mz de Marigorta, F. Palacios, J. Vicario
5-Ethoxy-1-(4-methoxyphenyl)-5-methyl-3-phenylimidazolidine-2,4-dione
MolBank,
2021;
M1218 - M1226
-
Ann-Katrine Jakobsen, Josephine Geertsen Keller, M. Gonzalez, E. Martin-Encinas, F. Palacios, C. Alonso, Birgitta R. Knudsen, Magnus Stougaard
A Dual-Sensor-Based Screening System for In Vitro Selection of TDP1 Inhibitors
Sensors,
2021;
21,
4832 - 4848
-
Xabier del Corte, Adrián López-Francés, Aitor Maestro, Ilia Villate-Beitia, Myriam Sainz-Ramos, Edorta Martínez de Marigorta, José Luis Pedraz, Francisco Palacios, Javier Vicario
A multicomponent protocol for the synthesis of highly functionalized gamma-lactam derivatives and their applications as antiproliferative agents
Pharmaceuticals,
2021;
14,
482 - 503
-
A. Selas, E. Martin-Encinas, M. Fuertes, C. Masdeu, C. Rubiales, F. Palacios, C. Alonso
A Patent review of topoisomerase I inhibitors (2016 – present)
Expert Opinion on Therapeutic Patents,
2021;
31,
473 - 508
-
Aitor Maestro, Xabier del Corte, Adrián López-Francés, Edorta Martinez de Marigorta, Francisco Palacios, Javier Vicario
Asymmetric Synthesis of Tetrasubstituted alpha-Aminophosphonic Acid Derivatives
Molecules,
2021;
26,
3202 - 3243
-
F. Palacios, A. M. Ochoa de Retana, J. M. de los Santos
Copper-catalyzed synthesis of aziridines
Copper in N-Heterocyclic Chemistry,
2021;
1 - 44 -
978-0-12-821263-9
-
A. Selas, G. Ramirez, , F. Palacios, C. Alonso
Design, synthesis and cytotoxic evaluation of diphenyl(quinolin-8-yl)phosphine oxides
Tetrahedron Letters,
2021;
70,
153019 - 153023
-
Xabier del Corte, Aitor Maestro, Edorta Martinez de Marigorta, Francisco Palacios, Javier Vicario
Enantioselective synthesis of unsaturated γ-lactams
Targets in heterocyclic systems. Chemistry and properties,
2021;
25,
22 - 52 -
9788886208758
-
E. Martin-Encinas, G. Rubiales, B. R. Knudssen, F. Palacios, C. Alonso
Fused chromeno and quinolino[1,8]naphthyridines: Synthesis and biological evaluation as topoisomerase I inhibitors and antiproliferative agents
Bioorganic Medicinal Chemistry,
2021;
40,
116177 - 116192
-
A. Selas M. Fuertes, E. Melcón-Fernández, Y. Pérez-Pertejo, R. M. Reguera, R. Balaña-Fouce,, B. R. Knudsen, F. Palacios, and C. Alonso
Hybrid Quinolinyl Phosphonates as Heterocyclic Carboxylate Isosteres: Synthesis and Biological Evaluation against Topoisomerase 1B (TOP1B)
Pharmaceuticals,
2021;
14,
784 - 908
-
Rizo-Liendo, Aitor, Iñigo Arberas-Jiménez, Endika Martin-Encinas, Ines Sifaoui, María Reyes-Batlle, Javier Chao-Pellicer, Concepción Alonso, Francisco Palacios, José E. Piñero, and Jacob Lorenzo-Morales.
Naphthyridine Derivatives Induce Programmed Cell Death in Naegleria fowleri
Pharnmaceuticals,
2021;
14,
1013 - 1028 -
ISSN: 1424-8247
-
Aitor Rizo-Liendo, Iñigo Arberas-Jiménez, Endika Martin-Encinas, Ines Sifaoui, María Reyes-Batlle, Javier Chao-Pellicer, Concepción Alonso, Francisco Palacios, José E. Piñero, Jacob Lorenzo-Morales
Naphthyridine Derivatives Induce Programmed Cell Death in Naegleria fowleri
Pharmaceuticals (1),
2021;
14,
1013 - 1028
-
M. Jewginski, K. Haremza , J. M. de los Santos , Z. Es Sbai, B. Oszywa, M. Pawelczak, F. Palacios, R. Latajka
Phosphinotripeptidic inhibitors of leucylaminopeptidases
International Journal of Molecular Sciences,
2021;
22,
5090 - 5117
-
Kamilla Vandsø Petersen, Asier Selas, Kirstine Mejlstrup Hymøller, Karol Mizielinski, Maria Thorsager, Magnus Stougaard, Conception Alonso, Francisco Palacios, Yolanda Perez Pertejo, Rosa Maria Reguera, Rafael Balana Fouce, Birgitta R. Knudsen, Cinzia Tesauro
Simple and Fast DNA Based Sensor System for Screening of Small-molecule compounds Targeting Eukaryotic Topoisomerase1
Pharmaceutics,
2021;
13 - 1255 -
1270
-
X. del Corte; A. López-Francés, E. Mz de Marigorta, F. Palacios, J. Vicario
Stereo- and regio-selective [3+3] annulation reaction catalyzed by ytterbium. Synthesis of bicyclic 1,4-dihydropyridines
Advanced Synthesis & Catalysis,
2021;
363,
0000 - 0000
-
V. Carramiñana, Ana M. Ochoa de Retana, F. Palacios, J M de los Santos
Synthesis and antiproliferative activity of phosphorus substituted 4-cyanooxazolines, 2-aminocyano oxazoliines, 2-iminocyanooxazolidines and 2-aminocyanothiazolines by rearrangement of cyanoaziridines
Molecules,
2021;
26,
4265 - 4292
-
A. López-Francés, X. del Corte; E. Mz de Marigorta, F. Palacios, J. Vicario
Ugi Reaction on alpha-Phosphorated Ketimines for the Synthesis of Tetrasubstituted alpha- Aminophosphonates and Their Applications as Antiproliferative Agents
Molecules,
2021;
26,
1654 - 1663
-
Maestro, A; Martínez de Marigorta, E. M.; Palacios, F.; Vicario, J.
alpha-Iminophosphonates: Useful Intermediates for Enantioselective Synthesis of alpha-Aminophosphonates
Asian Journal of Organic Chemistry,
2020;
9,
538 - 548
-
del Corte, X.; Lopez-Francés, A.; Maestro,A; de Marigorta, E. M; Palacios,F.; Vicario, J.
Bronsted Acid Catalyzed Multicomponent Synthesis of Phosphorus and Fluorine-Derived gamma-Lactam Derivatives
Journal of Organic Chemistry,
2020;
85,
14369 - 14383